(19)
(11) EP 1 235 815 A1

(12)

(43) Date of publication:
04.09.2002 Bulletin 2002/36

(21) Application number: 00976914.2

(22) Date of filing: 03.11.2000
(51) International Patent Classification (IPC)7C07D 239/84, C07D 403/12, A61K 31/517, C07D 239/78, C07D 239/80
(86) International application number:
PCT/US0030/376
(87) International publication number:
WO 0103/8315 (31.05.2001 Gazette 2001/22)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 22.11.1999 US 166840 P

(71) Applicant: WARNER-LAMBERT COMPANY
Morris PlainsNew Jersey 07950 (US)

(72) Inventors:
  • BARVIAN, Mark, Robert
    Ann Arbor, MI 48103 (US)
  • BATHINI, Yadagiri
    Edmonton, Alberta T6J 6W3 (CA)
  • DOBRUSIN, Ellen, Myra
    Ann Arbor, MI 48104 (US)
  • KALTENBRONN, James Stanley
    Ann Arbor, MI 48103 (US)
  • MICETICH, Ronald, George
    Sherwood Park, Alberta T8A 3V6 (CA)
  • SIDHU, Inderjit, S.
    Edmonton, Alberta T6L 2Y4 (CA)
  • SINGH, Rajeshwar
    Edmonton, Alberta T6K 1Z2 (CA)
  • TOOGOOD, Peter, Laurence
    Ann Arbor, MI 48108 (US)
  • WINTERS, Roy, Thomas
    Pinckney, MI 48169 (US)

(74) Representative: Tesch, Rudolf, Dr. et al
Warner-Lambert Company,c/o Gödecke GmbH,Patents
79090 Freiburg
79090 Freiburg (DE)

   


(54) QUINAZOLINES AND THEIR USE FOR INHIBITING CYCLIN-DEPENDENT KINASE ENZYMES