ACRYLOYL PEPTIDIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS - Patent 1242374

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EP 1 242 374 A1

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(43)	Date of publication:
	25.09.2002 Bulletin 2002/39

(21)	Application number: 00993255.9

(22)	Date of filing: 23.11.2000

(51)	International Patent Classification (IPC)⁷: C07D 207/34, C07D 403/14, A61P 35/02, A61K 31/40

(86)	International application number:
	PCT/EP0011/714

(87)	International publication number:
	WO 0104/0181 (07.06.2001 Gazette 2001/23)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

03.12.1999 GB 9928703

(71)	Applicant: Pharmacia & Italia S.p.A.
	20152 Milano (IT)

(72)	Inventors:
	COZZI, Paolo I-20133 Milan (IT) BERIA, Italo 20014 Nerviano (IT) CALDARELLI, Marina I-20147 Milan (IT) GERONI, Maria, Cristina, Rosa I-20149 Milan (IT) BARALDI, Pier, Giovanni I-44100 Ferrara (IT) ROMAGNOLI, Romeo I-44100 Ferrara (IT)

(74)	Representative: Longoni, Alessandra
	Pharmacia Italia S.p.A.,Patent Department,Viale Pasteur 10 20014 Nerviano (MI) 20014 Nerviano (MI) (IT)

(54)	ACRYLOYL PEPTIDIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS