A PROCESS FOR THE REGIOSELECTIVE SYNTHESIS OF 2,2-DIALKYL-4-SUBSTITUTED PIPERIDINES - Patent 1242377

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EP 1 242 377 A1

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(43)	Date of publication:
	25.09.2002 Bulletin 2002/39

(21)	Application number: 00982250.3

(22)	Date of filing: 06.12.2000

(51)	International Patent Classification (IPC)⁷: C07D 211/12, C07D 211/22, C07D 409/04

(86)	International application number:
	PCT/US0032/424

(87)	International publication number:
	WO 0104/6142 (28.06.2001 Gazette 2001/26)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

20.12.1999 US 172722 P

(71)	Applicant: ELI LILLY AND COMPANY
	Indianapolis, IN 46285 (US)

(72)	Inventor:
	HEATH, Perry, Clark Indianapolis, IN 46217 (US)

(74)	Representative: Vaughan, Jennifer Ann
	Eli Lilly and Company LimitedLilly Research CentreErl Wood Manor Windlesham, Surrey GU20 6PH Windlesham, Surrey GU20 6PH (GB)

(54)	A PROCESS FOR THE REGIOSELECTIVE SYNTHESIS OF 2,2-DIALKYL-4-SUBSTITUTED PIPERIDINES