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(11)

EP 1 246 823 A1

(12)

(43) Date of publication: 09.10.2002 Bulletin 2002/41 (21) Application number: 00990308.9 (22) Date of filing: 22.12.2000

(51) International Patent Classification (IPC)7: C07D 417/12, A61P 29/00, A61P 35/00, A61P 37/00, A61P 43/00, A61K 31/53, C07D 417/14, C07D 403/04, C07D 401/12, C07D 413/12, C07D 401/04, C07D 487/08, C07D 403/12 (86) International application number: PCT/US0035/049 (87) International publication number: WO 0104/7921 (05.07.2001 Gazette 2001/27)

(84) Designated Contracting States: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR Designated Extension States: AL LT LV MK RO SI (30) Priority: 28.12.1999 US 173227 P (71) Applicant: PHARMACOPEIA, INC. Princeton, NJ 08543 (US)	(72) Inventors: ERICKSON, Shawn, David Leonia, NJ 07605 (US) INGLESE, James Lansdale, PA 19446-1675 (US) LETOURNEAU, Jeffrey, John Princeton Junction, NJ 08550 (US) RIVIELLO, Christopher, Mark Yardley, PA 19067 (US) (74) Representative: Graf von Stosch, Andreas, Dr. rer. nat. et al Bosch - Graf v. Stosch - JehlePatentanwälteTheatinerstrasse 8 80333 München 80333 München (DE)