TOSYLPROLINE ANALOGS AS THYMIDYLATE SYNTHASE INHIBITORS - Patent 1252141

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EP 1 252 141 A1

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(43)	Date of publication:
	30.10.2002 Bulletin 2002/44

(21)	Application number: 01905352.9

(22)	Date of filing: 02.02.2001

(51)	International Patent Classification (IPC)⁷: C07D 207/48, C07D 211/96, A61K 31/445, A61K 31/401, A61P 31/04, A61P 31/12, A61P 33/00

(86)	International application number:
	PCT/US0103/391

(87)	International publication number:
	WO 0105/6987 (09.08.2001 Gazette 2001/32)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

02.02.2000 US 496378

(71)	Applicant: Sunesis Pharmaceuticals, Inc.
	San Francisco, CA 94080 (US)

(72)	Inventor:
	ERLANSON, Daniel, A. San Francisco, CA 94122 (US)

(74)	Representative: Hayes, Adrian Chetwynd et al
	Boult Wade Tennant,Verulam Gardens70 Gray's Inn Road London WC1X 8BT London WC1X 8BT (GB)

(54)	TOSYLPROLINE ANALOGS AS THYMIDYLATE SYNTHASE INHIBITORS