(19)
(11) EP 1 268 405 A1

(12)

(43) Date of publication:
02.01.2003 Bulletin 2003/01

(21) Application number: 01926512.3

(22) Date of filing: 02.04.2001
(51) International Patent Classification (IPC)7C07C 233/81, A61K 31/165
(86) International application number:
PCT/US0110/410
(87) International publication number:
WO 0107/4759 (11.10.2001 Gazette 2001/41)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 04.04.2000 US 542148

(71) Applicant: Allergan, Inc.
Irvine,California 92612 (US)

(72) Inventors:
  • NEHME, Alissar
    Newport Beach, CA 92660 (US)
  • BEARD, Richard, L.
    Newport Beach, CA 92660 (US)
  • CHANDRARATNA, Roshantha, A.
    Laguna Hills, CA 92653 (US)

(74) Representative: HOFFMANN - EITLE 
Patent- und RechtsanwälteArabellastrasse 4
81925 München
81925 München (DE)

   


(54) TREATMENT OF TUMORS WITH RAR ALPHA SELECTIVE RETINOID COMPOUNDS IN COMBINATION WITH OTHER ANTI-TUMOR AGENTS