(19)
(11) EP 1 268 454 A1

(12)

(43) Date of publication:
02.01.2003 Bulletin 2003/01

(21) Application number: 01924498.7

(22) Date of filing: 30.03.2001
(51) International Patent Classification (IPC)7C07D 295/18, C07D 317/58, C07D 213/38, C07D 239/42, C07D 241/20, C07D 401/04, C07D 211/58, C07D 405/04, C07D 211/60, C07D 211/22, C07D 211/42, C07D 211/26, A61K 31/506, A61P 25/28
(86) International application number:
PCT/US0110/297
(87) International publication number:
WO 0107/4796 (11.10.2001 Gazette 2001/41)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
LT LV RO SI

(30) Priority: 31.03.2000 US 193490 P

(71) Applicant: Bristol-Myers Squibb Pharma Company
Princeton,New Jersey 08543-4000 (US)

(72) Inventors:
  • THOMPSON, Lorin, Andrew
    Wilmington, DE 19809 (US)
  • KASIREDDY, Padmaja
    Kennett Square, PA 19348 (US)

(74) Representative: Howard, Paul Nicholas et al
Carpmaels & Ransford43 Bloomsbury Square
London WC1A 2RA
London WC1A 2RA (GB)

   


(54) SUCCINOYLAMINO HETEROCYCLES AS INHIBITORS OF A-BETA PROTEIN PRODUCTION