BIFUNCTIONAL INHIBITORS OF MALARIAL PROTEASES AND USES THEREOF - Patent 1274679

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EP 1 274 679 A1

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(43)	Date of publication:
	15.01.2003 Bulletin 2003/03

(21)	Application number: 01924983.8

(22)	Date of filing: 12.04.2001

(51)	International Patent Classification (IPC)⁷: C07C 317/00, A61K 31/00

(86)	International application number:
	PCT/US0112/000

(87)	International publication number:
	WO 0108/3433 (08.11.2001 Gazette 2001/45)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

21.04.2000 US 199023 P

(71)	Applicant: Enanta Pharmaceuticals, Inc.
	Cambridge, MA 02139 (US)

(72)	Inventor:
	ECKSTEIN, Jens, W. Arlington, MA 02476 (US)

(74)	Representative: Schlich, George William et al
	Mathys & SquireEuropean Patent Attorneys,100 Gray's Inn Road London WC1X 8AL London WC1X 8AL (GB)

(54)	BIFUNCTIONAL INHIBITORS OF MALARIAL PROTEASES AND USES THEREOF