(19)

(11)

EP 1 282 416 A2

(12)

(88) Date of publication A3: 12.09.2002 (43) Date of publication: 12.02.2003 Bulletin 2003/07 (21) Application number: 00986812.6 (22) Date of filing: 20.10.2000

(51) International Patent Classification (IPC)7: A61K 31/375, A61K 47/02, A61K 47/12, A01N 1/02 (86) International application number: PCT/US0041/407 (87) International publication number: WO 0108/9520 (29.11.2001 Gazette 2001/48)

(84) Designated Contracting States: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE Designated Extension States: AL LT LV MK RO SI (30) Priority: 19.05.2000 US 205870 P (71) Applicant: PROGENICS PHARMACEUTICALS, INC. Tarrytown, NY 10591 (US)	(72) Inventors: OLSON, William, C. Ossining, NY 10562 (US) ISRAEL, Robert, J. Livingston, NJ 07039 (US) BOYD, Thomas, A. Grandview, NY 10960 (US) (74) Representative: HOFFMANN - EITLE  Patent- und RechtsanwälteArabellastrasse 4 81925 München 81925 München (DE)