(19)
(11) EP 1 286 590 A2

(12)

(88) Date of publication A3:
27.12.2002

(43) Date of publication:
05.03.2003 Bulletin 2003/10

(21) Application number: 00976928.2

(22) Date of filing: 04.11.2000
(51) International Patent Classification (IPC)7A01N 37/18
(86) International application number:
PCT/US0030/416
(87) International publication number:
WO 0103/4631 (17.05.2001 Gazette 2001/20)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 05.11.1999 US 163911 P

(71) Applicant: Axonyx, Inc.
New York, NY 10022 (US)

(72) Inventor:
  • SOTO-JARA, Claudio
    CH-1287 Laconnex (CH)

(74) Representative: Wallace, Sheila Jane et al
Lloyd WiseCommonwealth House,1-19 New Oxford Street
London WC1A 1LW
London WC1A 1LW (GB)

   


(54) PEPTIDE ANALOGS AND MIMETICS SUITABLE FOR IN VIVO USE IN THE TREATMENT OF DISEASES ASSOCIATED WITH ABNORMAL PROTEIN FOLDING INTO AMYLOID, AMYLOID-LIKE DEPOSITS OR BETA-SHEET RICH PATHOLOGICAL PRECURSOR THEREOF