(19)
(11) EP 1 301 473 A2

(12)

(88) Date of publication A3:
30.01.2003

(43) Date of publication:
16.04.2003 Bulletin 2003/16

(21) Application number: 01954689.4

(22) Date of filing: 13.07.2001
(51) International Patent Classification (IPC)7C07C 271/22, C07K 1/107, C07K 19/00
(86) International application number:
PCT/US0122/194
(87) International publication number:
WO 0200/8245 (31.01.2002 Gazette 2002/05)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 13.07.2000 US 218113 P
29.09.2000 WO PCT/US00/26821
28.03.2001 US 279302 P
20.04.2001 US 839577

(71) Applicant: The Scripps Research Institute
La Jolla, CA 92037 (US)

(72) Inventors:
  • HAHN, Klaus, M.
    San Diego, CA 92131 (US)
  • TOUTCHKINE, Alexei
    San Diego, CA 92109 (US)
  • MUTHYALA, Rajeev
    Champaign, IL 61820 (US)
  • KRAYNOV, Vadim
    San Diego, CA 92121 (US)
  • BARK, Steven, J.
    San Diego, CA 92131 (US)
  • BURTON, Dennis, R.
    LaJolla, CA 92037 (US)
  • CHAMBERLAIN, Chester
    Cambridge,Massachusetts 02140 (US)

(74) Representative: Leifert & Steffan 
Patentanwälte,Burgplatz 21-22
40213 Düsseldorf
40213 Düsseldorf (DE)

   


(54) LABELED PEPTIDES, PROTEINS AND ANTIBODIES AND PROCESSES AND INTERMEDIATES USEFUL FOR THEIR PREPARATION