(19)
(11) EP 1 307 461 A2

(12)

(88) Date of publication A3:
18.07.2002

(43) Date of publication:
07.05.2003 Bulletin 2003/19

(21) Application number: 01958850.8

(22) Date of filing: 20.07.2001
(51) International Patent Classification (IPC)7C07D 495/04, A61K 31/407, A61P 29/00
// (C07D495/04, 333:00), C07D209:00
(86) International application number:
PCT/US0121/106
(87) International publication number:
WO 0201/2249 (14.02.2002 Gazette 2002/07)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 04.08.2000 US 223398 P

(71) Applicant: ELI LILLY AND COMPANY
Indianapolis, IN 46285 (US)

(72) Inventors:
  • BEIGHT, Douglas, Wade
    Frankfort, IN 46041 (US)
  • MORIN, John, Michael, Junior
    Brownsburg, IN 46112 (US)
  • SAWYER, Jason, Scott
    Indianapolis, IN 46220 (US)
  • SMITH, Edward, C., R.
    Fishers, IN 46038 (US)

(74) Representative: Kingsbury, Oliver William 
Eli Lilly and Company Limited,Erl Wood Manor,Sunninghill Road
Windlesham, Surrey GU20 6PH
Windlesham, Surrey GU20 6PH (GB)

   


(54) SUBSTITUTED PYRROLE COMPOUNDS AND THEIR USE AS SPLA2 INHIBITORS