(19)
(11) EP 1 313 705 A1

(12)

(43) Date of publication:
28.05.2003 Bulletin 2003/22

(21) Application number: 01968257.4

(22) Date of filing: 29.08.2001
(51) International Patent Classification (IPC)7C07D 213/74, C07D 401/12, C07D 213/73, C07D 471/04, A61K 31/4427, A61K 31/553, A61P 35/00, A61P 31/00
(86) International application number:
PCT/US0126/963
(87) International publication number:
WO 0201/8340 (07.03.2002 Gazette 2002/10)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 30.08.2000 US 229186 P

(71) Applicants:
  • Pharmacia Corporation
    St. Louis, MO 63167 (US)
  • Khanna, Ish Kumar
    Libertyville, IL 60048 (US)
  • Yu, Yi
    Skokie, IL 60077 (US)
  • Fun-Lu, Hwang
    Ballwin, MO 63021 (US)
  • Chandrakumar, Nizal S.
    Vernon Hills, IL 60061 (US)
  • Huff, Renee M.
    Park Ridge, IL 60068 (US)
  • Russell, Mark A.
    Gurnee, IL 60031 (US)
  • Boys, Mark L.
    Mt. Prospect, IL 60056 (US)
  • Schretzman, Lori A.
    Gurnee, IL 60031 (US)
  • Chen, Barbara B.
    Glenview, IL 60025 (US)
  • Desai, Bipinchandra N.
    Vernon Hills, IL 60061 (US)
  • Nagarajan, Srinivasan Raj
    Chesterfield, MO 63005 (US)
  • Gasiecki, Alan F.
    Vernon Hills, IL 60061 (US)
  • Penning, Thomas D.
    Elmhurst, IL 60126 (US)
  • Rogers, Thomas
    Ballwin, MO 63021 (US)
  • Wendt, John Adam
    Libertyville, IL 60048 (US)
  • Khilevich, Albert
    Buffalo Grove, IL 60089 (US)
  • Wang, Yaping
    Naperville, IL 60565 (US)

(72) Inventors:
  • KHANNA, Ish, Kumar
    Libertyville, IL 60048 (US)
  • YU, Yi
    Skokie, IL 60077 (US)
  • FUN-LU, Hwang
    Ballwin, MO 63021 (US)
  • CHANDRAKUMAR, Nizal, S.
    Vernon Hills, IL 60061 (US)
  • HUFF, Renee, M.
    Park Ridge, IL 60068 (US)
  • RUSSELL, Mark, A.
    Gurnee, IL 60031 (US)
  • BOYS, Mark, L.
    Mt. Prospect, IL 60056 (US)
  • SCHRETZMAN, Lori, A.
    Gurnee, IL 60031 (US)
  • CHEN, Barbara, B.
    Glenview, IL 60025 (US)
  • DESAI, Bipinchandra, N.
    Vernon Hills, IL 60061 (US)
  • NAGARAJAN, Srinivasan, Raj
    Chesterfield, MO 63005 (US)
  • GASIECKI, Alan, F.
    Vernon Hills, IL 60061 (US)
  • PENNING, Thomas, D.
    Elmhurst, IL 60126 (US)
  • ROGERS, Thomas
    Ballwin, MO 63021 (US)
  • WENDT, John, Adam
    Libertyville, IL 60048 (US)
  • KHILEVICH, Albert
    Buffalo Grove, IL 60089 (US)
  • WANG, Yaping
    Naperville, IL 60565 (US)
  • DEVADAS, Balekudra
    Chesterfield, MO 63017 (US)

(74) Representative: Albrecht, Thomas, Dr. et al
Kraus & Weisert,Thomas-Wimmer-Ring 15
80539 München
80539 München (DE)

   


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