(19)
(11) EP 1 322 652 A1

(12)

(43) Date of publication:
02.07.2003 Bulletin 2003/27

(21) Application number: 01975165.0

(22) Date of filing: 13.09.2001
(51) International Patent Classification (IPC)7C07D 498/04
(86) International application number:
PCT/US0126/023
(87) International publication number:
WO 0202/4705 (28.03.2002 Gazette 2002/12)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 22.09.2000 US 234649 P

(71) Applicant: ELI LILLY AND COMPANY
Indianapolis, Indiana 46285 (US)

(72) Inventors:
  • BARNETT, Charles, Jackson
    Indianapolis, IN 46240 (US)
  • GU, Rui Lin
    Indianapolis, IN 46236 (US)
  • KOBIERSKI, Michael, Edward
    Greenwood, IN 46142 (US)

(74) Representative: Burnside, Ivan John et al
Eli Lilly and Company LimitedEuropean Patent OperationsErl Wood ManorSunninghill Road
Windlesham, Surrey GU20 6PH
Windlesham, Surrey GU20 6PH (GB)

   


(54) STEREOSELECTIVE PROCESS FOR PREPARING CYCLOHEXYL AMINE DERIVATIVES