(19)
(11) EP 1 324 985 A1

(12)

(43) Date of publication:
09.07.2003 Bulletin 2003/28

(21) Application number: 01979912.1

(22) Date of filing: 28.09.2001
(51) International Patent Classification (IPC)7C07D 209/12, A61K 31/4045
(86) International application number:
PCT/US0142/389
(87) International publication number:
WO 0202/8831 (11.04.2002 Gazette 2002/15)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 02.10.2000 US 237241 P

(71) Applicant: Merck & Co., Inc.
Rahway,New Jersey 07065-0907 (US)

(72) Inventors:
  • TROTTER, B., Wesley
    Rahway, NJ 07065-0907 (US)
  • QUIGLEY, Amy, G.
    Rahway, NJ 07065-0907 (US)
  • DINSMORE, Christopher, J.
    Rahway, NJ 07065-0907 (US)
  • LUMMA, William, C., Jr.
    Rahway, NJ 07065-0907 (US)
  • SISKO, John, T.
    Rahway, NJ 07065-0907 (US)

(74) Representative: Horgan, James Michael Frederic et al
Merck & Co., Inc.,Terlings Park,Eastwick Road
Harlow,Essex CM20 2QR
Harlow,Essex CM20 2QR (GB)

   


(54) INHIBITORS OF PRENYL-PROTEIN TRANSFERASE