(19)
(11) EP 1 345 901 A2

(12)

(88) Date of publication A3:
23.01.2003

(43) Date of publication:
24.09.2003 Bulletin 2003/39

(21) Application number: 01974983.7

(22) Date of filing: 15.08.2001
(51) International Patent Classification (IPC)7C07D 211/90
(86) International application number:
PCT/NL0100/601
(87) International publication number:
WO 0205/3535 (11.07.2002 Gazette 2002/28)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 29.12.2000 US 258613 P
16.03.2001 US 809351

(71) Applicant: Bioorganics B.V.
6545 CM Nijmegen (NL)

(72) Inventors:
  • PETERS, Theodorus, Hendricus, Antonius
    NL-6814 JB Arnhem (NL)
  • BENNEKER, Franciscus, Bernardus, Gemma
    NL-6991 HA Rheden (NL)
  • SLANINA, Pavel
     (CZ)
  • BARTL, Jiri
    664 47 Strelice (CZ)

(74) Representative: Prins, Hendrik Willem 
Arnold & Siedsma,Advocaten en Octrooigemachtigden,Sweelinckplein 1
2517 GK Den Haag
2517 GK Den Haag (NL)

   


(54) PROCESS FOR MAKING AMLODIPINE, DERIVATIVES THEREOF, AND PRECURSORS THEREFOR