(19)
(11) EP 1 355 637 A2

(12)

(88) Date of publication A3:
21.08.2003

(43) Date of publication:
29.10.2003 Bulletin 2003/44

(21) Application number: 01944426.4

(22) Date of filing: 12.06.2001
(51) International Patent Classification (IPC)7A61K 31/00
(86) International application number:
PCT/US0118/773
(87) International publication number:
WO 0109/7794 (27.12.2001 Gazette 2001/52)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

(30) Priority: 21.06.2000 US 213073 P

(71) Applicant: GEORGETOWN UNIVERSITY MEDICAL CENTER
Washington, DC 20007 (US)

(72) Inventors:
  • LIN, Chen-Yong
    Falls Church, VA 22043 (US)
  • DICKSON, Robert, B.
    Kensington, MD 20845 (US)
  • WANG, Shaomeng,University of Michigan
    Ann Arbor, Michigan 48109-0934 (US)
  • ENYEDY, Istvan
    Mount Ranier, MD 20712 (US)
  • LEE, Sheau-Ling
    Falls Church, VA 22042 (US)

(74) Representative: Daniels, Jeffrey Nicholas et al
Page White & Farrer54 Doughty Street
London WC1N 2LS
London WC1N 2LS (GB)

   


(54) INHIBITORS OF MATRIPTASE FOR THE TREATMENT OF CANCER