(19)
(11) EP 1 355 698 A2

(12)

(88) Date of publication A3:
31.07.2003

(43) Date of publication:
29.10.2003 Bulletin 2003/44

(21) Application number: 01980019.2

(22) Date of filing: 10.10.2001
(51) International Patent Classification (IPC)7A61P 3/10, A61P 5/50, A61K 31/655, A61K 31/195, A61K 31/185
// (C07C311/47, 309:51)
(86) International application number:
PCT/US0142/733
(87) International publication number:
WO 0203/0514 (18.04.2002 Gazette 2002/16)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 11.10.2000 US 239636 P

(71) Applicant: TELIK, INC.
Palo Alto, CA 94304 (US)

(72) Inventors:
  • MANCHEM, Prasad V. V. S. V.
    South San Francisco, CA 94080 (US)
  • LUM, Robert, T.
    Palo Alto, CA 94306 (US)
  • SCHOW, Steven, R.
    Redwood City, CA 94065 (US)

(74) Representative: Barz, Peter, Dr. 
PatentanwaltKaiserplatz 2
80803 München
80803 München (DE)

   


(54) INSULIN RECEPTOR ACTIVATORS FOR THE TREATMENT OF METABOLIC DISORDERS IN HUMANS RESULTING FROM TREATMENT OF HIV INFECTION WITH HIV PROTEASE INHIBITORS