N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD - Patent 1373192

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EP 1 373 192 A1

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(43)	Date of publication:
	02.01.2004 Bulletin 2004/01

(21)	Application number: 02707042.4

(22)	Date of filing: 18.03.2002

(51)	International Patent Classification (IPC)⁷: C07C 235/82, C07C 255/60, C07D 231/56, C07D 311/74, C07C 323/40, C07D 307/79, C07D 213/40, C07D 215/12, C07D 319/20, C07D 317/52, A61K 31/195, A61K 31/335, A61K 31/41, A61K 31/435, A61P 15/00

(86)	International application number:
	PCT/IB2002/000807

(87)	International publication number:
	WO 2002/079143 (10.10.2002 Gazette 2002/41)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

28.03.2001 GB 0107750
30.05.2001 GB 0113112
17.08.2001 GB 0120152

(71)	Applicants:
	Pfizer Limited Sandwich,Kent CT13 9NJ (GB) GB PFIZER INC. New York, N.Y. 10017 (US) AT BE CH CY DE DK ES FI FR GR IE IT LU MC NL PT SE TR LI

(72)	Inventors:
	CHALLENGER, Stephen Sandwich,Kent CT13 9NJ (GB) COOK, Andrew Simon Sandwich,Kent CT13 9NJ (GB) GILLMORE, Adam Thomas Sandwich,Kent CT13 9NJ (GB) MIDDLETON, Donald Stuart Sandwich,Kent CT13 9NJ (GB) PRYDE, David Cameron Sandwich,Kent CT13 9NJ (GB) STOBIE, Alan Sandwich,Kent CT13 9NJ (GB)

(74)	Representative: Rutt, Jason Edward et al
	U.K. Patent DepartmentPfizer LimitedRamsgate Road Sandwich, Kent CT13 9NJ Sandwich, Kent CT13 9NJ (GB)

(54)	N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD