(19)
(11) EP 1 373 307 A2

(12)

(88) Date of publication A3:
24.07.2003

(43) Date of publication:
02.01.2004 Bulletin 2004/01

(21) Application number: 02757911.9

(22) Date of filing: 01.04.2002
(51) International Patent Classification (IPC)7C07K 14/00, C07K 11/00, C12N 9/00
(86) International application number:
PCT/US2002/010116
(87) International publication number:
WO 2002/079223 (10.10.2002 Gazette 2002/41)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 31.03.2001 US 280624 P

(71) Applicant: BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM
Austin, TX 78701 (US)

(72) Inventors:
  • PAUL, Sudhir
    Missouri City, TX 77459 (US)
  • NISHIYAMA, Yasuhiro
    Houston, TX 77059 (US)

(74) Representative: Cripps, Joanna Elizabeth et al
Mewburn EllisYork House23 Kingsway
London WC2B 6HP
London WC2B 6HP (GB)

   


(54) COVALENTLY REACTIVE TRANSITION STATE ANALOGS AND METHODS OF USE THEREOF