(19)
(11) EP 1 377 580 A2

(12)

(88) Date of publication A3:
12.09.2003

(43) Date of publication:
07.01.2004 Bulletin 2004/02

(21) Application number: 02703087.3

(22) Date of filing: 17.01.2002
(51) International Patent Classification (IPC)7C07D 487/04
(86) International application number:
PCT/US2002/000502
(87) International publication number:
WO 2002/060871 (08.08.2002 Gazette 2002/32)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 30.01.2001 US 264996 P

(71) Applicant: ELI LILLY AND COMPANY
Indianapolis, Indiana 46285 (US)

(72) Inventors:
  • FILLA, Sandra, Ann
    Franklin, IN 46131 (US)
  • FLAUGH, Michael, Edward
    Indianapolis, IN 46256 (US)
  • GILLIG, James, Ronald
    Indianapolis, IN 46268 (US)
  • HEINZ, Lawrence, Joseph
    Pittsboro, IN 46167 (US)
  • KRUSHINSKI, Joseph, Herman, Junior
    Brownburg, IN 46112 (US)
  • LIU, Bin
    Fishers, IN 46038 (US)
  • PINEIRO-NUNEZ, Marta, Maria
    Brownsburg, IN 46112 (US)
  • SCHAUS, John, Mehnert
    Zionsville, IN 46077 (US)
  • WARD, John, Stanley
    Redwood City, CA 94065 (US)

(74) Representative: Kingsbury, Oliver William et al
Eli Lilly and Company Limited,Erl Wood Manor,Sunninghill Road
Windlesham, Surrey GU20 6PH
Windlesham, Surrey GU20 6PH (GB)

   


(54) BENZENESULFONIC ACID INDOL-5-YL ESTERS AS ANTAGONISTS OF THE 5-HT6 RECEPTOR