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<ep-patent-document id="EP02780964B8W1" file="EP02780964W1B8.xml" lang="en" country="EP" doc-number="1389203" kind="B8" correction-code="W1" date-publ="20100310" status="c" dtd-version="ep-patent-document-v1-4">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIE......FI....CY..TR................................................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  2999001/0</B007EP></eptags></B000><B100><B110>1389203</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20100310</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>02780964.9</B210><B220><date>20020226</date></B220><B240><B241><date>20030925</date></B241><B242><date>20050224</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>271941 P</B310><B320><date>20010227</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20100310</date><bnum>201010</bnum></B405><B430><date>20040218</date><bnum>200408</bnum></B430><B450><date>20091202</date><bnum>200949</bnum></B450><B452EP><date>20090605</date></B452EP><B480><date>20100310</date><bnum>201010</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 403/04        20060101AFI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 209/48        20060101ALI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/454       20060101ALI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/4035      20060101ALI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/402       20060101ALI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/513       20060101ALI20031024BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P  43/00        20060101ALI20031024BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>ANALOGA VON THALIDOMID ALS  ANGIOGENESEINHIBITOREN</B542><B541>en</B541><B542>ANALOGS OF THALIDOMIDE AS  ANGIOGENESIS INHIBITORS</B542><B541>fr</B541><B542>ANALOGUES DE THALIDOMIDE UTILISES COMME INHIBITEURS  DE L'ANGIOGENESE</B542></B540><B560><B561><text>EP-A- 0 856 513</text></B561><B561><text>WO-A-94/20085</text></B561><B561><text>WO-A-97/37988</text></B561><B561><text>WO-A-98/03502</text></B561><B562><text>GÜTSCHOW M ET AL: "Aza analogues of thalidomide: synthesis and evaluation as inhibitors of tumor necrosis factor-alpha production in vitro." BIOORGANIC &amp; MEDICINAL CHEMISTRY. ENGLAND APR 2001, vol. 9, no. 4, April 2001 (2001-04), pages 1059-1065, XP002207264 ISSN: 0968-0896</text></B562><B562><text>TEUBERT U ET AL: "5'-SUBSTITUTED THALIDOMIDE ANALOGS AS MODULATORS OF TNF-ALPHA*" ARCHIV DER PHARMAZIE, VCH VERLAGSGESELLSCHAFT MBH, WEINHEIM, DE, vol. 331, no. 1, 1998, pages 7-12, XP002072713 ISSN: 0365-6233</text></B562></B560></B500><B700><B720><B721><snm>FIGG, William, D.</snm><adr><str>10451 Breckinridge Lane</str><city>Fairfax, VA 22030</city><ctry>US</ctry></adr></B721><B721><snm>EGER, Kurt</snm><adr><str>Alte Landstrasse 15/4</str><city>72072 Tuebingen</city><ctry>DE</ctry></adr></B721><B721><snm>TEUBERT, Uwe</snm><adr><str>Berliner Strasse 3a</str><city>31789 Hameln</city><ctry>DE</ctry></adr></B721><B721><snm>WEISS, Michael</snm><adr><str>Dorfstrasse 21</str><city>06571 Wiehe-Garnbach</city><ctry>DE</ctry></adr></B721><B721><snm>GUETSCHOW, Michael,
Pharmazeutisches Institut</snm><adr><str>Universitaet Bonn,
Kreuzbergweg 26</str><city>53115 Bonn</city><ctry>DE</ctry></adr></B721><B721><snm>HECKER, Thomas</snm><adr><str>Richard-Breslau Strasse 6</str><city>99094 Erfurt</city><ctry>DE</ctry></adr></B721><B721><snm>HAUSCHILDT, Sunna</snm><adr><str>Pistorisstrasse 19</str><city>04229 Leipzig</city><ctry>DE</ctry></adr></B721></B720><B730><B731><snm>The Government of the United States of America, 
represented by The Secretary Department of Health 
and Human services</snm><iid>04038490</iid><irf>FB12903/E18024E</irf><adr><str>Office of Technology Transfer 
Suite 325, 6011 Executive Blvd.</str><city>Rockville, MD 20852</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Gowshall, Jonathan Vallance</snm><iid>00061534</iid><adr><str>Forrester &amp; Boehmert 
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