(19)
(11) EP 1 390 740 A1

(12)

(43) Date of publication:
25.02.2004 Bulletin 2004/09

(21) Application number: 02739334.7

(22) Date of filing: 23.05.2002
(51) International Patent Classification (IPC)7G01N 31/00, G01N 33/566, C07H 17/00
(86) International application number:
PCT/US2002/016218
(87) International publication number:
WO 2002/095391 (28.11.2002 Gazette 2002/48)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 24.05.2001 US 293362 P

(71) Applicant: Endacea, Inc.
Research Triangle Park, NC 27709-2076 (US)

(72) Inventor:
  • WILSON, Constance, Neely
    Research Triangle Park, NC 27709 (US)

(74) Representative: Horner, Martin Grenville et al
Cruikshank & Fairweather19 Royal Exchange Square
Glasgow G1 3AEScotland
Glasgow G1 3AEScotland (GB)

   


(54) METHODS AND FORMULATIONS FOR INCREASING THE AFFINITY OF A 1? ADENOSINE RECEPTOR LIGANDS FOR THE A 1? ADENOSINE RECEPTOR