(19)
(11) EP 1 392 657 A2

(12)

(88) Date of publication A3:
13.11.2003

(43) Date of publication:
03.03.2004 Bulletin 2004/10

(21) Application number: 01275089.9

(22) Date of filing: 19.11.2001
(51) International Patent Classification (IPC)7C07D 223/08
(86) International application number:
PCT/US2001/051647
(87) International publication number:
WO 2003/053331 (03.07.2003 Gazette 2003/27)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 22.11.2000 US 252508 P

(71) Applicant: SmithKline Beecham Corporation
King of Prussia, PA 19406 (US)

(72) Inventors:
  • MARQUIS, Robert, W., Jr.
    King of Prussia, PA 19406 (US)
  • VEBER, Daniel, F.
    King of Prussia, PA 19406 (US)
  • YAMASHITA, Dennis, S.
    King of Prussia, PA 19406 (US)

(74) Representative: Rutter, Keith et al
GlaxoSmithKlineCorporate Intellectual Property (CN9.25.1)980 Great West Road
Brentford, Middlesex TW8 9GS
Brentford, Middlesex TW8 9GS (GB)

   


(54) PROTEASE INHIBITORS