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<ep-patent-document id="EP02774050B8W1" file="EP02774050W1B8.xml" lang="en" country="EP" doc-number="1399424" kind="B8" correction-code="W1" date-publ="20081001" status="c" dtd-version="ep-patent-document-v1-3">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESI....FI....CY..TR............................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  2999001/0</B007EP></eptags></B000><B100><B110>1399424</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20081001</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>02774050.5</B210><B220><date>20020522</date></B220><B240><B241><date>20031210</date></B241><B242><date>20040423</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>0112812</B310><B320><date>20010525</date></B320><B330><ctry>GB</ctry></B330></B300><B400><B405><date>20081001</date><bnum>200840</bnum></B405><B430><date>20040324</date><bnum>200413</bnum></B430><B450><date>20080709</date><bnum>200828</bnum></B450><B452EP><date>20080117</date></B452EP><B480><date>20081001</date><bnum>200840</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 223/22        20060101AFI20021211BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/55        20060101ALI20021211BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61P  25/08        20060101ALI20021211BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>VERFAHREN ZUR HERSTELLUNG VON 10,11 DIHYDRO 10 HYDROXY 5H-DIBENZ/B,F/AZEPIN-5-CARBONSÄUREAMID UND 10,11 DIHYDRO 10 OXO-5H-DIBENZ/B,F/AZEPIN-5 CARBONSÄUREAMID</B542><B541>en</B541><B542>METHOD FOR PREPARATION OF 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE AND 10,11-DIHYDRO-10-0X0-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE</B542><B541>fr</B541><B542>PROCEDE DE PREPARATION DU 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE ET DU 10,11-DIHYDRO-10-0X0-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE</B542></B540><B560><B561><text>CH-A- 642 950</text></B561><B561><text>DE-A- 2 246 842</text></B561><B561><text>NL-A- 7 902 811</text></B561><B561><text>US-A- 5 753 646</text></B561><B562><text>K.M. BAKER, J. CSETENYI, A. FRIGERIO, P.L. MORSELLI: "a metabolite of carbamazepine" J. OF MED. CHEMISTRY, vol. 16, no. 6, 1973, pages 703-705, XP002209649 cited in the application</text></B562><B562><text>CANALI L ET AL: "Synthesis of resins with pendently-bound chiral manganese-salen complexes and use as heterogeneous asymmetric alkene epoxidation catalysts" REACTIVE &amp; FUNCTIONAL POLYMERS, ELSEVIER SCIENCE PUBLISHERS BV, NL, vol. 40, no. 2, 15 May 1999 (1999-05-15), pages 155-168, XP004164106 ISSN: 1381-5148</text></B562><B562><text>SENANAYAKE C H ET AL: "The Role of 4-(3-Phenylpropyl)pyridine N-Oxide (P3NO) in the Manganese-Salen-Catalyzed Asymmetric Epoxidation of Indene" TETRAHEDRON LETTERS, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, vol. 37, no. 19, 6 May 1996 (1996-05-06), pages 3271-3274, XP004029376 ISSN: 0040-4039</text></B562><B562><text>G. BELLUCCI, G. BERTI, C. CHIAPPE, A.LIPPI, F. MARIONI: "the metabolism of carbamazepine in Humans" J. MED.CHEM, vol. 30, 1987, pages 768-773, XP002209650 cited in the application</text></B562><B562><text>M. OSHIMA, H. YAMAZAKI, I. SHIMIZU, M. NISAR, J. TSUJI: "Palladium-Catalyzed selective hydrogenolysis of alkenyloxiranes with formic acid." J.AM.CHEM.SOC, vol. 111, 1989, pages 6280-6287, XP002209651</text></B562><B562><text>E.J. COREY: " a new Cr(IV) reagent for the catalytic oxidation of secundary alcohols" TETRAHEDRON LETTERS, vol. 26, no. 48, 1985, pages 5855-5858, XP001095121</text></B562><B562><text>GRANT S M ET AL: "OXCARBAZEPINE. A REVIEW OF ITS PHARMACOLOGY AND THERAPEUTIC POTENTIAL IN EPILEPSY, TRIGEMINAL NEURALGIA AND AFFECTIVE DISORDERS" DRUGS, ADIS INTERNATIONAL LTD, AT, vol. 43, no. 6, 1992, pages 873-888, XP002039768 ISSN: 0012-6667 cited in the application</text></B562><B562><text>BENES J ET AL: "Anticonvulsant and Sodium Channel-Blocking Properties of Novel 10,11-Dihydro-5H-dibenz[b,f]azepine-5-carb oxamide Derivatives" JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, vol. 42, 1999, pages 2582-2587, XP002206156 ISSN: 0022-2623 cited in the application</text></B562><B562><text>S.-I. MURAHASHI, T. NAOTA, Y. ODA, N. HIRAI: "Ruthenium catalysed oxidation of Alcohols with peracids" SYNLETT, vol. 7, 1995, XP001093973</text></B562></B560></B500><B600><B620EP><parent><cdoc><dnum><anum>08075527.5</anum><pnum>1958938</pnum></dnum><date>20080602</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>LEARMONTH, David, Alexander</snm><adr><str>Rua Adelino Amaro da Costa, 109-2oE,
Vermoin</str><city>P-4470-225 Maia</city><ctry>PT</ctry></adr></B721></B720><B730><B731><snm>BIAL - Portela &amp; Ca., S.A.</snm><iid>08349740</iid><irf>PAC/20714 EP</irf><adr><city>Av. da Siderurgia Nacional
4745-457 S. Mamede do Coronado - Trofa</city><ctry>PT</ctry></adr></B731></B730><B740><B741><snm>Curtis, Philip Anthony</snm><sfx>et al</sfx><iid>00055274</iid><adr><str>A.A. Thornton &amp; Co. 
235 High Holborn</str><city>London WC1V 7LE</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry><ctry>TR</ctry></B840><B844EP><B845EP><ctry>SI</ctry><date>20031210</date></B845EP></B844EP><B860><B861><dnum><anum>GB2002002356</anum></dnum><date>20020522</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2002096881</pnum></dnum><date>20021205</date><bnum>200249</bnum></B871></B870><B880><date>20040324</date><bnum>200413</bnum></B880></B800></SDOBI>
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