(19)
(11) EP 1 401 427 A2

(12)

(88) Date of publication A3:
20.03.2003

(43) Date of publication:
31.03.2004 Bulletin 2004/14

(21) Application number: 02739712.4

(22) Date of filing: 05.06.2002
(51) International Patent Classification (IPC)7A61K 31/341, A61K 31/443, A61K 31/497, C07D 307/58, C07D 405/10
(86) International application number:
PCT/US2002/017846
(87) International publication number:
WO 2002/098363 (12.12.2002 Gazette 2002/50)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 06.06.2001 US 295812 P
29.06.2001 US 301868 P

(71) Applicant: Agouron Pharmaceuticals, Inc.
La Jolla, CA 92037 (US)

(72) Inventors:
  • SUN, Eric, T.
    San Diego, CA 92130 (US)
  • ANDERSON, Mark, B.
    Orinda, CA 94563 (US)
  • ANDERES, Kenna, Lynn
    San Diego, CA 92130 (US)
  • CHRISTIE, Lance, Christopher
    Vista, CA 92083 (US)
  • DO, Quyen-Quyen, Thuy
    San Diego, CA 92131 (US)
  • FENG, Jun
    Carlsbad, CA 92009 (US)
  • GOETZEN, Thomas
    San Diego, CA 92115 (US)
  • HONG, Yufeng
    San Diego, CA 92128 (US)
  • KRAYNOV, Eugenia, Anatolievna
    San Diego, CA 92121 (US)
  • LI, Haitao
    San Diego, CA 92130 (US)
  • LUTHIN, David, Robert
    Encinitas, CA 92024 (US)
  • PADERES, Genevieve, D.
    San Diego, CA 92121 (US)
  • PATHAK, Ved, P.
    San Diego, CA 92130 (US)
  • RAJAPAKSE, Ranjan, Jagath
    Poway, CA 92064 (US)
  • SHACKELFORD, Scott
    Escondido, CA 92029 (US)
  • TOMPKINS, Eileen, Valenzuela
    Escondido, CA 92026 (US)
  • TRUESDALE, Larry, Kenneth
    San Diego, CA 92131 (US)
  • VAZIR, Haresh
    Salinas, CA 93905 (US)

(74) Representative: Tesch, Rudolf, Dr. et al
c/o Pfizer GmbH,Arzneimittelwerk GödeckeMooswaldallee 1
79090 Freiburg
79090 Freiburg (DE)

   


(54) NON-PEPTIDE GNRH AGENTS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR THEIR USES, AND PROCESSES FOR PREPARING THEM