(19)
(11) EP 1 404 680 A2

(12)

(88) Date of publication A3:
08.01.2004

(43) Date of publication:
07.04.2004 Bulletin 2004/15

(21) Application number: 01271082.8

(22) Date of filing: 22.10.2001
(51) International Patent Classification (IPC)7C07D 493/04
(86) International application number:
PCT/US2001/051428
(87) International publication number:
WO 2002/067239 (29.08.2002 Gazette 2002/35)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 24.10.2000 US 242822 P

(71) Applicant: GLAXO GROUP LIMITED
Greenford, Middlesex UB6 ONN (GB)

(72) Inventors:
  • DAVIS, Roman,GlaxoSmithKline
    Research Triangle Park, NC 27709 (US)
  • LOVELACE, Thomas Claiborne,GlaxoSmithKline
    Research Triangle Park, NC 27709 (US)

(74) Representative: Crawley, Karen Anne et al
GlaxoSmithKlineCorporate Intellectual Property (CN9.25.1)980 Great West Road
Brentford, Middlesex TW8 9GS
Brentford, Middlesex TW8 9GS (GB)

   


(54) PROCESS FOR PREPARING INTERMEDIATES OF HIV PROTEASE INHIBITORS