(19)
(11) EP 1 409 512 A1

(12)

(43) Date of publication:
21.04.2004 Bulletin 2004/17

(21) Application number: 01946642.4

(22) Date of filing: 21.06.2001
(51) International Patent Classification (IPC)7C07J 13/00, A61K 31/57, A61P 5/28
(86) International application number:
PCT/US2001/019889
(87) International publication number:
WO 2002/000681 (03.01.2002 Gazette 2002/01)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

(30) Priority: 27.06.2000 US 214561 P
14.05.2001 US 290881 P

(71) Applicant: Aventis Pharma S.A.
92160 Antony (FR)

(72) Inventors:
  • PEET, Norton, P.
    North Andover, MA 01845 (US)
  • WEINTRAUB, Philip, M.
    Warren, NJ 07059 (US)
  • BURKHART, Joseph, P.
    Plainfield, IN 46168 (US)
  • GATES, Cynthia, A.
    Cambridge, MA 02140 (US)

   


(54) 20-FLUORO-17(20)-VINYL STEROIDS AS INHIBITORS OF C17-20-LYASE AND 5-ALPHA REDUCTASE