(19)
(11) EP 1 423 119 A1

(12)

(43) Date of publication:
02.06.2004 Bulletin 2004/23

(21) Application number: 02731761.9

(22) Date of filing: 10.05.2002
(51) International Patent Classification (IPC)7A61K 31/4995, A61K 31/5365, C07C 57/58, C07C 59/68, C07C 233/65, C07C 235/46, C07D 471/08, C07D 471/18, C07D 498/18
(86) International application number:
PCT/US2002/014966
(87) International publication number:
WO 2002/089806 (14.11.2002 Gazette 2002/46)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 10.05.2001 US 289828 P

(71) Applicant: Agouron Pharmaceuticals, Inc.
La Jolla, CA 92037 (US)

(72) Inventors:
  • GUO, Chuangxing
    San Diego, CA 92130 (US)
  • AUGELLI-SZAFRAN, Corinne, E.
    Ann Arbor, MI 48103 (US)
  • BARTA, Nancy, Sue
    Brighton, MI 48116 (US)
  • BENDER, Steven, Lee
    Oceanside, CA 92054 (US)
  • BIGGE, Christopher, Franklin
    Ann Arbor, MI 48105 (US)
  • CAPRATHE, Bradley, William
    Livonia, MI 48154 (US)
  • CHATTERJEE, Arindam
    Fishers, IN 46038 (US)
  • DEAL, Judith
    Wildomar, CA 92595 (US)
  • DONG, Liming
    San Diego, CA 92126 (US)
  • FAY, Lorraine, Kathleen
    Upsilanti, MI 48198 (US)
  • HOU, Xinjun
    San Diego, CA 92129 (US)
  • HUDACK, Raymond, Andrew, Jr.
    Grand Blanc, MI 48439 (US)

(74) Representative: Tesch, Rudolf, Dr. 
c/o Pfizer GmbH,Arzneimittelwerk GödeckeMooswaldallee 1
79090 Freiburg
79090 Freiburg (DE)

   


(54) HETEROBICYCLES FKBP-LIGANDS