(19)
(11) EP 1 423 411 A2

(12)

(88) Date of publication A3:
25.09.2003

(43) Date of publication:
02.06.2004 Bulletin 2004/23

(21) Application number: 02744537.8

(22) Date of filing: 02.07.2002
(51) International Patent Classification (IPC)7C07K 5/072, A61K 38/05, A61P 25/00
(86) International application number:
PCT/US2002/019825
(87) International publication number:
WO 2003/006489 (23.01.2003 Gazette 2003/04)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 09.07.2001 EP 01500175
23.11.2001 EP 01500275

(71) Applicant: ELI LILLY AND COMPANY
Indianapolis, Indiana 46285 (US)

(72) Inventors:
  • BUENO MELENDO, Ana, Belen
    28100 Alcobendas (ES)
  • DE DIOS, Alfonso
    28100 Alcobendas (ES)
  • DOMINGUEZ-FERNANDEZ, Carmen
    28100 Alcobendas (ES)
  • FERRITTO CRESPO, Rafael
    28100 Alcobendas (ES)
  • HERIN, Marc,Lilly MSG Dev. Centre S. A.
    B-1348 Mont-Sai (BE)
  • MARTIN, Jose, Alfredo
    28100 Alcobendas (ES)
  • MARTIN-CABREJAS, Luisa, Maria
    28100 Alcobendas (ES)
  • MARTINEZ-GRAU, Maria, Angeles
    28100 Alcobendas (ES)
  • MASSEY, Steven, Marc
    Indianapolis, IN 46268 (US)
  • MONN, James, Allen
    Indianapolis, IN 46268 (US)
  • MONTERO SALGADO, Carlos
    28100 Alcobendas (ES)
  • PEDREGAL-TERCERO, Concepcion
    28100 Alcobendas (ES)
  • VALLI, Matthew, John
    Zionsville, IN 46077 (US)

(74) Representative: Kingsbury, Oliver William 
Eli Lilly and Company Limited,European Patent Operations,Lilly Research Centre,Sunninghill Road
Windlesham,Surrey GU20 6PH
Windlesham,Surrey GU20 6PH (GB)

   


(54) PRODRUGS OF EXCITATORY AMINO ACIDS