NEW GENERATION TRIPLE-TARGETING, CHIRAL, BROAD-SPECTRUM ANTIMICROBIAL 7-SUBSTITUTED PIPERIDINO-QUINOLONE CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, COMPOSITIONS AND USE AS MEDICAMENTS - Patent 1453824

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EP 1 453 824 A1

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(43)	Date of publication:
	08.09.2004 Bulletin 2004/37

(21)	Application number: 02796957.5

(22)	Date of filing: 12.12.2002

(51)	International Patent Classification (IPC)⁷: C07D 401/04, C07D 413/04, A61P 31/04, A61K 31/47

(86)	International application number:
	PCT/IN2002/000232

(87)	International publication number:
	WO 2003/050107 (19.06.2003 Gazette 2003/25)

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR IE IT LI LU MC NL PT SE SI SK TR
	Designated Extension States:
	AL LT LV MK RO

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Priority:

13.12.2001 US 341165 P
23.04.2002 US 128996
24.04.2002 WO PCT/IN02/00111

(71)	Applicants:
	Wockhardt Limited Mumbai 400 051,Maharashtra (IN) Patel, Mahesh V. Bandra (E),400 051 Mumbai (IN) Deshpande, Prasad K. Bandra (E),400 051 Mumbai (IN) Agarwal, Shiv Kumar Bandra (E),400 051 Mumbai (IN) Chugh, Yati Bandra (E),400 051 Mumbai (IN) Shukla, Milind C. Bandra (E),400 051 Mumbai (IN)

(72)	Inventors:
	DE SOUZA, Noel J.Wockhardt Limited Bandra(E), 400 051 Mumbai (IN) PATEL, MaheshWockhardt Limited Bandra(E), 400 051 Mumbai (IN) DESHPANDE, Prasad Wockhardt Limited Bandra(E), 400 051 Mumbai (IN) AGARWAL,Shiv Kumar Wockhardt Limited Bandra(E), 400 051 Mumbai (IN) CHUGH, Yati Wockhardt Limited Bandra(E), 400 051 Mumbai (IN) SHUKLA, Milind Wockhardt Limited Bandra(E), 400 051 Mumbai (IN)

(74)	Representative: Ebner von Eschenbach, Jennifer et al
	Ladas & Parry,Dachauerstrasse 37 80335 München 80335 München (DE)

(54)	NEW GENERATION TRIPLE-TARGETING, CHIRAL, BROAD-SPECTRUM ANTIMICROBIAL 7-SUBSTITUTED PIPERIDINO-QUINOLONE CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, COMPOSITIONS AND USE AS MEDICAMENTS