(19)
(11) EP 1 480 999 A2

(12)

(88) Date of publication A3:
25.03.2004

(43) Date of publication:
01.12.2004 Bulletin 2004/49

(21) Application number: 03743123.6

(22) Date of filing: 07.02.2003
(51) International Patent Classification (IPC)7C07K 5/023, C07K 5/027, A61K 38/05, A61P 9/10, A61P 19/02, A61P 25/28
(86) International application number:
PCT/US2003/003987
(87) International publication number:
WO 2003/072528 (04.09.2003 Gazette 2003/36)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT SE SI SK TR
Designated Extension States:
AL LT LV MK RO

(30) Priority: 08.02.2002 US 355390 P

(71) Applicant: Idun Pharmaceuticals
San Diego, CA 92121 (US)

(72) Inventors:
  • KARANEWSKY, Donald, S.
    Escondido, CA 92029 (US)
  • KALISH, Vincent, J.
    Annapolis, MD 21401 (US)
  • ROBINSON, Edard, D.
    San Diego, CA 92122 (US)
  • ULLMAN, Brett, R.
    San Diego, CA 92103 (US)

(74) Representative: Grünecker, Kinkeldey, Stockmair & SchwanhäusserAnwaltssozietät 
Maximilianstrasse 58
80538 München
80538 München (DE)

   


(54) (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES