(19)
(11) EP 1 482 939 A1

(12)

(43) Date of publication:
08.12.2004 Bulletin 2004/50

(21) Application number: 02729099.8

(22) Date of filing: 01.05.2002
(51) International Patent Classification (IPC)7: A61K 31/445, C07D 405/12
(86) International application number:
PCT/US2002/013826
(87) International publication number:
WO 2003/072104 (04.09.2003 Gazette 2003/36)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 22.02.2002 US 358916 P

(71) Applicant: TEVA PHARMACEUTICAL INDUSTRIES LTD.
49131 Petah Tiqva (IL)

(72) Inventors:
  • PILARSKI, Gideon
    58487 Holon (IL)
  • AVRUTOV, Ilya
    42842 Bat Hefer (IL)

(74) Representative: Gallagher, Kirk James et al
D Young & Co120 Holborn
London EC1N 2DY
London EC1N 2DY (GB)

   


(54) PREPARATION OF PAROXETINE INVOLVING NOVEL INTERMEDIATES