PROPARGYLAMINO INDAN DERIVATIVES AND PROPARGYLAMINO TETRALIN DERIVATIVES AS BRAIN-SELECTIVE MAO INHIBITORS - Patent 1490324

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EP 1 490 324 A2

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(88)	Date of publication A3:
	31.12.2003

(43)	Date of publication:
	29.12.2004 Bulletin 2004/53

(21)	Application number: 03716197.3

(22)	Date of filing: 27.02.2003

(51)	International Patent Classification (IPC)⁷: C07C 211/00, C07C 261/00, C07C 269/00, C07C 271/00, A01N 33/02, A01N 47/10, A61K 31/27, A61K 31/135

(86)	International application number:
	PCT/US2003/005871

(87)	International publication number:
	WO 2003/072055 (04.09.2003 Gazette 2003/36)

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT SE SI SK TR
	Designated Extension States:
	AL LT LV MK RO

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Priority:

27.02.2002 US 85674

(71)	Applicant: TEVA PHARMACEUTICAL INDUSTRIES LTD.
	49131 Petah Tiqva (IL)

(72)	Inventors:
	BLAUGRUND, Eran 76449 Rehovot (IL) HERZIG, Yaacov 43266 R'ananna (IL) STERLING, Jeffrey Jerusalem 97275 (IL)

(74)	Representative: Almond-Martin, Carol et al
	Ernest Gutmann - Yves Plasseraud S.A.3, rue Chauveau-Lagarde 75008 Paris 75008 Paris (FR)

(54)	PROPARGYLAMINO INDAN DERIVATIVES AND PROPARGYLAMINO TETRALIN DERIVATIVES AS BRAIN-SELECTIVE MAO INHIBITORS