(19)
(11) EP 1 513 808 A2

(12)

(88) Date of publication A3:
22.04.2004

(43) Date of publication:
16.03.2005 Bulletin 2005/11

(21) Application number: 03756085.1

(22) Date of filing: 23.05.2003
(51) International Patent Classification (IPC)7C07D 207/08, C07D 205/04, C07D 211/38, A61K 31/40, A61K 31/397, A61K 31/445, A61P 3/10, C12Q 1/37
(86) International application number:
PCT/IB2003/002257
(87) International publication number:
WO 2003/101958 (11.12.2003 Gazette 2003/50)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 04.06.2002 US 386157 P

(71) Applicant: Pfizer Products Inc.
Groton,Connecticut 06340 (US)

(72) Inventors:
  • HULIN, BernardPfizer Global Research and Develop.
    Groton, CT 06340 (US)
  • PARKER, J. CatherinePfizer Global Research &Dev.
    Groton, CT 06340 (US)

(74) Representative: Laurent, Claire et al
PFIZER PGRDEuropean Pharma Patent Dept.23/25 Avenue du Docteur Lannelongue
75668 Paris Cedex 14
75668 Paris Cedex 14 (FR)

   


(54) FLUORINATED CYCLIC AMIDES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS