(19)
(11) EP 1 524 979 A2

(12)

(88) Date of publication A3:
27.05.2004

(43) Date of publication:
27.04.2005 Bulletin 2005/17

(21) Application number: 03743752.2

(22) Date of filing: 31.07.2003
(51) International Patent Classification (IPC)7: A61K 31/427, C07D 417/06, C07D 493/04, C07D 207/40, C07C 323/24, A61K 47/48
(86) International application number:
PCT/EP2003/008483
(87) International publication number:
WO 2004/012735 (12.02.2004 Gazette 2004/07)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 31.07.2002 DE 10234975
07.02.2003 DE 10305098
05.03.2003 US 451673 P

(71) Applicant: Schering AG
13353 Berlin (DE)

(72) Inventors:
  • BERGER, Markus
    13347 Berlin (DE)
  • SIEMEISTER, Gerhard
    13503 Berlin (DE)
  • KLAR, Ulrich
    13503 Berlin (DE)
  • WILLUDA, Jörg
    13156 Berlin (DE)
  • MENRAD, Andreas
    16515 Oranienburg (DE)
  • BOSSLET, Klaus
    13465 Berlin (DE)

   


(54) NEW EFFECTOR CONJUGATES, PROCESS FOR THEIR PRODUCTION AND THEIR PHARMACEUTICAL USE