METHODS FOR THE SYNTHESIS OF SUBSTITUTED PURINES - Patent 1529048

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EP 1 529 048 A2

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(88)	Date of publication A3:
	03.03.2005

(43)	Date of publication:
	11.05.2005 Bulletin 2005/19

(21)	Application number: 02801053.6

(22)	Date of filing: 12.10.2002

(51)	International Patent Classification (IPC)⁷: C07D 473/16, C07D 473/40, C07D 473/18

(86)	International application number:
	PCT/US2002/032679

(87)	International publication number:
	WO 2003/031405 (17.04.2003 Gazette 2003/16)

(84)	Designated Contracting States:
	AT BE BG CH CY CZ DE DK EE ES FI FR GB GR IE IT LI LU MC NL PT SE SK TR
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

12.10.2001 US 328741 P
07.01.2002 US 346552 P
08.01.2002 US 347037 P

(71)	Applicants:
	IRM LLC Hamilton HM LX (BM) The Scripps Research Institute La Jolla, CA 92037 (US)

(72)	Inventors:
	DING, Sheng San Diego, CA 92122 (US) DING, Qiang San Diego, CA 92122 (US) GRAY, Nathanael, S. San Diego, CA 92122 (US) SCHULTZ, Peter, G. La Jolla, CA 92037 (US)

(74)	Representative: Woods, Geoffrey Corlett
	J.A. KEMP & CO.Gray's Inn14 South Square London WC1R 5JJ London WC1R 5JJ (GB)

(54)	METHODS FOR THE SYNTHESIS OF SUBSTITUTED PURINES