(19)
(11) EP 1 534 239 A2

(12)

(88) Date of publication A3:
26.08.2004

(43) Date of publication:
01.06.2005 Bulletin 2005/22

(21) Application number: 03811294.2

(22) Date of filing: 04.08.2003
(51) International Patent Classification (IPC)7A61K 9/00, A61K 9/127, A61K 9/14
(86) International application number:
PCT/US2003/024353
(87) International publication number:
WO 2004/054500 (01.07.2004 Gazette 2004/27)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 05.08.2002 US 213352
17.09.2002 US 246802

(71) Applicant: BAXTER INTERNATIONAL INC.
Deerfield, Illinois 60015 (US)

(72) Inventors:
  • WERLING, Jane
    Arlington Heights, IL 60005 (US)
  • KIPP, James, E.
    Wauconda, IL 60084 (US)
  • SRIRAM, Rajaram
    Glenview, IL 60025 (US)
  • DOTY, Mark, J.
    Grayslake, IL 60030 (US)
  • REBBECK, Christine, L.
    Algonquin, IL 60102 (US)
  • WONG, Joseph, Chung, Tak
    Gurnee, IL 60031 (US)

(74) Representative: Dee, Ian Mark et al
Eric Potter Clarkson,Park View House,58 The Ropewalk
Nottingham NG1 5DD
Nottingham NG1 5DD (GB)

   


(54) PREPARATION OF SUBMICRON SIZED PARTICLES WITH POLYMORPH CONTROL AND NEW POLYMORPH OF ITRACONAZOLE