| (84) |
Designated Contracting States: |
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AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR |
| (30) |
Priority: |
07.08.2002 US 401693 P
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| (43) |
Date of publication of application: |
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08.06.2005 Bulletin 2005/23 |
| (73) |
Proprietors: |
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- Novartis AG
4056 Basel (CH) Designated Contracting States: BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
- Novartis Pharma GmbH
1230 Wien (AT) Designated Contracting States: AT
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| (72) |
Inventor: |
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- MC KENNA, Jeffrey
San Diego, CA 92111 (US)
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| (74) |
Representative: de Weerd, Petrus G.W. et al |
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Novartis International AG
Corporate Intellectual Property 4002 Basel 4002 Basel (CH) |
| (56) |
References cited: :
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- YAMAUCHI, MASAHIGE ET AL: "Reactivity of 2,4(5)-dialkylimidazoles. Synthesis of 6,7,8,9-tetrahydro-
5H-imidazo[1,5-a][1,4]diazepine derivatives" CHEMICAL & PHARMACEUTICAL BULLETIN (1976),
24(7), 1480-4 , XP009019004
- YAMAUCHI, MASASHIGE ET AL: "Synthesis of 6,7,8,9-tetrahydro-5H-imidazo[1,5-a][1,4]d
iazepines" CHEMISTRY & INDUSTRY (LONDON, UNITED KINGDOM) (1976), (1), 31-2 , XP009019005
- JANIN Y L ET AL: "Imidazo[1,5-g][1,4]diazepines, TIBO Analogues Lacking the Phenyl
Ring: Synthesis and Evaluation as Anti-HIV Agents" TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS,
AMSTERDAM, NL, vol. 52, no. 48, 25 November 1996 (1996-11-25), pages 15157-15170,
XP004105102 ISSN: 0040-4020
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