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<ep-patent-document id="EP03784194B8W1" file="EP03784194W1B8.xml" lang="en" country="EP" doc-number="1537114" kind="B8" correction-code="W1" date-publ="20071003" status="c" dtd-version="ep-patent-document-v1-1">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESI....FIRO..CY..TRBGCZEEHU..SK................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>DIM360 (Ver 1.5  21 Nov 2005) -  2999001/0</B007EP><B070EP>The file contains technical information submitted after the application was filed and not included in this specification</B070EP><B078EP><date>20070510</date></B078EP></eptags></B000><B100><B110>1537114</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20071003</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>03784194.7</B210><B220><date>20030806</date></B220><B240><B241><date>20050307</date></B241><B242><date>20050621</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>401693 P</B310><B320><date>20020807</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20071003</date><bnum>200740</bnum></B405><B430><date>20050608</date><bnum>200523</bnum></B430><B450><date>20060809</date><bnum>200632</bnum></B450><B452EP><date>20060113</date></B452EP><B472><B475><date>20060809</date><ctry>BE</ctry><date>20060809</date><ctry>IT</ctry></B475></B472><B480><date>20071003</date><bnum>200740</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 487/04        20060101AFI20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/519       20060101ALI20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/5517      20060101ALI20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61P   5/40        20060101ALI20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C07D 487/04        20060101ALN20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>C07D 241/00        20060101ALN20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>C07D 235/00        20060101ALN20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>C07D 487/04        20060101ALN20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>C07D 243/00        20060101ALN20040302BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 235/00        20060101ALN20040302BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>ORGANISCHE VERBINDUNGEN ALS MITTEL ZUR BEHANDLUNG VON ALDOSTERONBEDINGTEN ZUSTÄNDEN</B542><B541>en</B541><B542>ORGANIC COMPOUNDS AS AGENTS FOR THE TREATMENT OF ALDOSTERONE MEDIATED CONDITIONS</B542><B541>fr</B541><B542>COMPOSES ORGANIQUES SERVANT D'AGENTS POUR LE TRAITEMENT D'ETATS PATHOLOGIQUES INDUITS PAR L'ALDOSTERONE</B542></B540><B560><B561><text>WO-A-97/00257</text></B561><B562><text>YAMAUCHI, MASAHIGE ET AL: "Reactivity of 2,4(5)-dialkylimidazoles. Synthesis of 6,7,8,9-tetrahydro- 5H-imidazo[1,5-a][1,4]diazepine derivatives" CHEMICAL &amp; PHARMACEUTICAL BULLETIN (1976), 24(7), 1480-4 , XP009019004</text></B562><B562><text>YAMAUCHI, MASASHIGE ET AL: "Synthesis of 6,7,8,9-tetrahydro-5H-imidazo[1,5-a][1,4]d iazepines" CHEMISTRY &amp; INDUSTRY (LONDON, UNITED KINGDOM) (1976), (1), 31-2 , XP009019005</text></B562><B562><text>JANIN Y L ET AL: "Imidazo[1,5-g][1,4]diazepines, TIBO Analogues Lacking the Phenyl Ring: Synthesis and Evaluation as Anti-HIV Agents" TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, vol. 52, no. 48, 25 November 1996 (1996-11-25), pages 15157-15170, XP004105102 ISSN: 0040-4020</text></B562></B560></B500><B700><B720><B721><snm>MC KENNA, Jeffrey</snm><adr><str>4695 Mount Bigelow</str><city>San Diego, CA 92111</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>Novartis AG</snm><iid>02240429</iid><irf>PC/4-32611A/USN</irf><adr><str>Lichtstrasse 35</str><city>4056 Basel</city><ctry>CH</ctry></adr><B736EP><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B736EP></B731><B731><snm>Novartis Pharma GmbH</snm><iid>04273610</iid><irf>PC/4-32611A/USN</irf><adr><str>Brunner Strasse 59</str><city>1230 Wien</city><ctry>AT</ctry></adr><B736EP><ctry>AT</ctry></B736EP></B731></B730><B740><B741><snm>de Weerd, Petrus G.W.</snm><sfx>et al</sfx><iid>00092224</iid><adr><str>Novartis International AG 
Corporate Intellectual Property</str><city>4002 Basel</city><ctry>CH</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B860><B861><dnum><anum>EP2003008720</anum></dnum><date>20030806</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2004014914</pnum></dnum><date>20040219</date><bnum>200408</bnum></B871></B870><B880><date>20050608</date><bnum>200523</bnum></B880></B800></SDOBI>
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