(19)
(11) EP 1 539 781 A2

(12)

(88) Date of publication A3:
11.03.2004

(43) Date of publication:
15.06.2005 Bulletin 2005/24

(21) Application number: 03760343.8

(22) Date of filing: 12.06.2003
(51) International Patent Classification (IPC)7C07H 17/00
(86) International application number:
PCT/US2003/018734
(87) International publication number:
WO 2003/105766 (24.12.2003 Gazette 2003/52)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 12.06.2002 US 388006 P
24.02.2003 US 449553 P

(71) Applicant: UNIVERSITY OF VIRGINIA PATENT FOUNDATION
Charlottesville,Virginia 22903 (US)

(72) Inventors:
  • SMITH, Jeffrey, A.
    Earlysville, VA 22936 (US)
  • LANNIGAN-MACARA, Deborah, A.
    Charlottesville, VA 22903 (US)
  • POTEET-SMITH, Celeste, E.
    Earlysville, VA 22936 (US)
  • HECHT, Sidney, M.
    Charlottesville, VA 22911 (US)
  • XU, Yaming
    Charlottesville, VA 22901 (US)
  • BRAUTIGAN, David, L.
    Charlottesville, VA 22901 (US)

(74) Representative: Richards, William John et al
D Young & Co,120 Holborn
London EC1N 2DY
London EC1N 2DY (GB)

   


(54) RSK INHIBITORS AND THERAPEUTIC USES THEREOF