(19)
(11) EP 1 558 599 A2

(12)

(88) Date of publication A3:
29.07.2004

(43) Date of publication:
03.08.2005 Bulletin 2005/31

(21) Application number: 03779296.7

(22) Date of filing: 24.10.2003
(51) International Patent Classification (IPC)7C07D 401/04, A61K 31/4523
(86) International application number:
PCT/US2003/034002
(87) International publication number:
WO 2004/041777 (21.05.2004 Gazette 2004/21)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 30.10.2002 US 422447 P

(71) Applicant: Merck & Co., Inc.
Rahway,New Jersey 07065-0907 (US)

(72) Inventors:
  • GOBLE, Stephen, D.
    Rahway, NJ 07065-0907 (US)
  • PASTERNAK, Alexander
    Rahway, NJ 07065-0907 (US)
  • YANG, Lihu
    Rahway, NJ 07065-0907 (US)

(74) Representative: Man, Jocelyn et al
Merck & Co.,Inc.,European Patent Department,Terlings Park,Eastwick Road
Harlow,Essex CM20 2QR
Harlow,Essex CM20 2QR (GB)

   


(54) HETEROARYLPIPERIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY