(19)
(11) EP 1 567 494 A1

(12)

(43) Date of publication:
31.08.2005 Bulletin 2005/35

(21) Application number: 03739242.0

(22) Date of filing: 17.06.2003
(51) International Patent Classification (IPC)7C07D 211/26, C07D 401/10, C07D 211/46, C07D 211/62, C07D 471/10, C07D 401/04, C07D 401/12
(86) International application number:
PCT/US2003/019601
(87) International publication number:
WO 2004/050623 (17.06.2004 Gazette 2004/25)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 02.12.2002 WO PCT/US02/38480

(71) Applicant: Ortho-McNeil Pharmaceutical, Inc.
Raritan, NJ 08869-0602 (US)

(72) Inventors:
  • APODACA, Richard
    San Diego, CA 92108 (US)
  • DENG, Xiaohu
    San Diego, CA 92129 (US)
  • JABLOBNOWSKI, Jill, A.
    San Diego, CA 92129 (US)
  • MANI, Neelakandha
    San Diego, CA 92129 (US)
  • PANDIT, Chennagiri, R.
    San Diego, CA 92129 (US)
  • XIAO, Wei
    San Diego, CA 92130 (US)

(74) Representative: Fisher, Adrian John et al
CARPMAELS & RANSFORD 43-45 Bloomsbury Square
London WC1A 2RA
London WC1A 2RA (GB)

   


(54) METHODS FOR PREPARING PHENYLALKYNE DERIVATIVES