(19)
(11) EP 1 569 641 A2

(12)

(88) Date of publication A3:
08.07.2004

(43) Date of publication:
07.09.2005 Bulletin 2005/36

(21) Application number: 03787112.6

(22) Date of filing: 20.11.2003
(51) International Patent Classification (IPC)7: A61K 31/428, C07D 277/82
(86) International application number:
PCT/US2003/037592
(87) International publication number:
WO 2004/047756 (10.06.2004 Gazette 2004/24)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 21.11.2002 US 301540

(71) Applicant: Teva Pharmaceutical Industries Limited
Petah Tikvah 49131 (IL)

(72) Inventors:
  • STERLING, Jeffrey
    Jerusalem 97275 (IL)
  • HAYARDENY, Liat
    Tel-Aviv 69391 (IL)
  • FALB, Eliezer
    Givataim 53450 (IL)
  • HERZIG, Yaacov
    Raanana 43266 (IL)
  • LERNER, David
    Jerusalem 97241 (IL)
  • BLAUGRUND, Eran
    Rehovot 76449 (IL)

(74) Representative: Nachshen, Neil Jacob et al
D Young & Co 120 Holborn
London EC1N 2DY
London EC1N 2DY (GB)

   


(54) PROPARGYL-TRIFLUOROMETHOXY-AMINO-BENZOTHIAZOLE DERIVATIVES