(19)
(11) EP 1 569 645 A2

(12)

(88) Date of publication A3:
02.09.2004

(43) Date of publication:
07.09.2005 Bulletin 2005/36

(21) Application number: 03813364.1

(22) Date of filing: 09.12.2003
(51) International Patent Classification (IPC)7A61K 31/44
(86) International application number:
PCT/US2003/039166
(87) International publication number:
WO 2004/054505 (01.07.2004 Gazette 2004/27)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 12.12.2002 US 432807 P

(71) Applicant: Pharmacia Corporation
Chesterfield, MO 63017-1732 (US)

(72) Inventors:
  • REINHARD, Emily, J.
    Ridgewood, NJ 07450 (US)
  • KOLODZIEJ, Stephen, A.
    Ballwin, MO 63021 (US)
  • ANDERSON, David, R.
    Lake St. Louis, MO 63367 (US)
  • STEHLE, Nathan, W.
    Grafton, WI 53024 (US)
  • VERNIER, William, F.
    Oceanside, CA 92056 (US)
  • LEE, Len, F.
    St. Charles, MO 63303 (US)
  • HEGDE, Shridhar, G.
    Ballwin, MO 63021 (US)

(74) Representative: Albrecht, Thomas 
Kraus & Weisert, Thomas-Wimmer-Ring 15
80539 München
80539 München (DE)

   


(54) METHOD OF USING AMINOCYANOPYRIDINE COMPOUNDS AS MITOGEN ACTIVATED PROTEIN KINASE-ACTIVATED PROTEIN KINASE-2 INHIBITORS