(19)
(11) EP 1 572 615 B8

(12) CORRECTED EUROPEAN PATENT SPECIFICATION
Note: Bibliography reflects the latest situation

(15) Correction information:
Corrected version no 1 (W1 B1)

(48) Corrigendum issued on:
14.07.2010 Bulletin 2010/28

(45) Mention of the grant of the patent:
17.03.2010 Bulletin 2010/11

(21) Application number: 03782373.9

(22) Date of filing: 11.12.2003
(51) International Patent Classification (IPC): 
C07D 207/16(2006.01)
(86) International application number:
PCT/EP2003/014082
(87) International publication number:
WO 2004/052817 (24.06.2004 Gazette 2004/26)

(54)

PROCESS FOR THE SYNTHESIS OF PEPTIDES CONTAINING A 4-HYDORXY-PROLINE SUBSTRUCTURE

PROZESS FÜR DIE HERSTELLUNG VON PEPTIDEN, DIE EINE 4-HYDORXY-PROLIN SUBSTRUKTUR ENTHALTEN

PROCEDE DE SYNTHESE PEPTIDIQUE CONTENANT UNE SOUS-STRUCTURE DE 4-HYDROXY-PROLINE

(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR

(30) Priority: 12.12.2002 GB 0229020
16.12.2002 GB 0229280

(43) Date of publication of application:
14.09.2005 Bulletin 2005/37

(73) Proprietors:
  • Novartis AG
    4056 Basel (CH)
    Designated Contracting States:
    LU IT IE HU GR GB FR FI ES EE DK DE CZ CY LI CH BG BE PT NL MC RO SE SI SK TR 
  • Novartis Pharma GmbH
    1230 Wien (AT)
    Designated Contracting States:
    AT 

(72) Inventors:
  • WIETFELD, Bernhard
    79588 Efringen-Kirchen (DE)
  • PRIKOSZOVICH, Walter
    CH-4124 Schönenbuch (CH)
  • ERB, Dr. Bernhard
    5073 Gipf-Oberfrick (CH)
  • PACHINGER, Werner
    4057 Basel (CH)


(56) References cited: : 
WO-A-02/10192
DE-A- 4 306 839
 WO-A-97/01579
   
  • W.M. BANDARANAYAKE ET.AL.: "ANOMALOUS ACETOXYLATION OF AROMATIC NUCLEI: SOME STRUCTURAL REQUIREMENTS IN THE SUBSTRATE" AUST. J. CHEM., vol. 34, no. 1, 1981, pages 115-129, XP009029409
  • W. WALTER: "Beyer Walter LEHRBUCH DER ORGANISCHEN CHEMIE" 1988 , S. HIRZEL VERLAG , STUTTGART XP002277902 PAGE 188, PARAGRAPH 2.20.2.2. page 188, line 4 - line 11
  • D. HELLWINKEL ET.AL.: "Tieffarbige, durchkonjugierte Multi-Triphenylmethykium-Ionen" ANGEW. CHEM., vol. 99, no. 8, 1987, pages 822-823, XP009029552
   
Note: Within nine months from the publication of the mention of the grant of the European patent, any person may give notice to the European Patent Office of opposition to the European patent granted. Notice of opposition shall be filed in a written reasoned statement. It shall not be deemed to have been filed until the opposition fee has been paid. (Art. 99(1) European Patent Convention).