(19)
(11) EP 1 603 885 A1

(12)

(43) Date of publication:
14.12.2005 Bulletin 2005/50

(21) Application number: 04717503.9

(22) Date of filing: 04.03.2004
(51) International Patent Classification (IPC)7C07D 231/54, C07D 401/06, C07D 401/04, C07D 403/10, C07D 401/12, C07D 403/12, C07D 403/14, C07D 401/14, C07D 405/14, C07D 417/14, C07D 405/12, C07D 417/12, C07D 403/04, A61K 31/416, A61P 35/00
(86) International application number:
PCT/US2004/006921
(87) International publication number:
WO 2004/080973 (23.09.2004 Gazette 2004/39)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
Designated Extension States:
AL LT LV MK

(30) Priority: 07.03.2003 US 384325
03.03.2004 US 792564

(71) Applicant: ABBOTT LABORATORIES
Abbott Park,Illinois 60064-6008 (US)

(72) Inventors:
  • TONG, Yunsong
    Grayslake, IL 60030 (US)
  • CLAIBORNE, Akiyo, K.
    Mundelein, IL 60060 (US)
  • LI, Gaoquan
    Park City, IL 60085 (US)
  • LIN, Nan-Horng
    Vernon Hills, IL 60061 (US)
  • SHAM, Hing
    Vernon Hills, IL 60061 (US)
  • TAO, Zhi-Fu
    Gurnee, IL 60031 (US)
  • SOWIN, Tom
    Wadsworth, IL 60083 (US)

(74) Representative: Modiano, Micaela Nadia et al
Modiano, Josif, Pisanty & Staub Ltd., Baaderstrasse 3
80469 München
80469 München (DE)

   


(54) FUSED TRI AND TETRA-CYCLIC PYRAZOLE KINASE INHIBITORS