<?xml version="1.0" encoding="UTF-8"?>
<!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.5//EN" "ep-patent-document-v1-5.dtd">
<ep-patent-document id="EP05012130B8W1" file="EP05012130W1B8.xml" lang="en" country="EP" doc-number="1604676" kind="B8" correction-code="W1" date-publ="20161214" status="c" dtd-version="ep-patent-document-v1-5">
<SDOBI lang="en"><B000><eptags><B001EP>......DE....FRGB....................................................................................</B001EP><B005EP>J</B005EP><B007EP>JDIM360 Ver 1.28 (29 Oct 2014) -  2999001/0</B007EP></eptags></B000><B100><B110>1604676</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20161214</date></B140><B150><B151>W1</B151><B153>54</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>05012130.0</B210><B220><date>20050606</date></B220><B240><B241><date>20060519</date></B241><B242><date>20080130</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>2004168996</B310><B320><date>20040607</date></B320><B330><ctry>JP</ctry></B330><B310>2004169052</B310><B320><date>20040607</date></B320><B330><ctry>JP</ctry></B330></B300><B400><B405><date>20161214</date><bnum>201650</bnum></B405><B430><date>20051214</date><bnum>200550</bnum></B430><B450><date>20161102</date><bnum>201644</bnum></B450><B452EP><date>20160429</date></B452EP><B480><date>20161214</date><bnum>201650</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C12N   9/02        20060101AFI20160322BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>Aromatase Transkriptionsaktivatorenextrakte</B542><B541>en</B541><B542>Aromatase transcription activators extracts</B542><B541>fr</B541><B542>Extraits comprenant des activateurs de transcription de l'aromatase</B542></B540><B560><B561><text>EP-A- 1 338 283</text></B561><B561><text>WO-A-00/13661</text></B561><B561><text>US-A1- 2004 265 399</text></B561><B562><text>HARADA NOBUHIRO ET AL: "Unique regulation of expression of human aromatase in the placenta." THE JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY. SEP 2003, vol. 86, no. 3-5, September 2003 (2003-09), pages 327-334, XP002342087 ISSN: 0960-0760</text></B562><B562><text>HARADA N: "Aberrant expression of aromatase in breast cancer tissues." THE JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY. APR 1997, vol. 61, no. 3-6, April 1997 (1997-04), pages 175-184, XP002342088 ISSN: 0960-0760</text></B562><B562><text>MORINAGA HIDETAKA ET AL: "A benzimidazole fungicide, benomyl, and its metabolite, carbendazim, induce aromatase activity in a human ovarian granulose-like tumor cell line (KGN)." ENDOCRINOLOGY. APR 2004, vol. 145, no. 4, April 2004 (2004-04), pages 1860-1869, XP002342089 ISSN: 0013-7227</text></B562><B562><text>ZAVA D T ET AL: "ESTROGEN AND PROGESTIN BIOACTIVITY OF FOODS, HERBS, AND SPICES (44247)" PROCEEDINGS OF THE SOCIETY FOR EXPERIMENTAL BIOLOGY &amp; MEDICINE, ACADEMIC PRESS INC. NEW YORK, US, vol. 217, no. 3, 1998, pages 369-378, XP008026916 ISSN: 0037-9727</text></B562><B562><text>CHEN S ET AL: "Modulation of aromatase expression in human breast tissue." THE JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY. DEC 2001, vol. 79, no. 1-5, December 2001 (2001-12), pages 35-40, XP002342090 ISSN: 0960-0760</text></B562><B562><text>JEONG H J ET AL: "Aromatase inhibitors from Isodon excisus var. coreanus." ARCHIVES OF PHARMACAL RESEARCH. JUN 2000, vol. 23, no. 3, June 2000 (2000-06), pages 243-245, XP008051234 ISSN: 0253-6269</text></B562><B562><text>LEE TAE-KYUN ET AL: "Inhibitory effects of Scutellaria barbata D. Don. and Euonymus alatus Sieb. on aromatase activity of human leiomyomal cells." IMMUNOPHARMACOLOGY AND IMMUNOTOXICOLOGY. AUG 2004, vol. 26, no. 3, August 2004 (2004-08), pages 315-327, XP008051235 ISSN: 0892-3973</text></B562><B562><text>HUANG BU-MIIN ET AL: "Upregulation of steroidogenic enzymes and ovarian 17beta-estradiol in human granulosa-lutein cells by Cordyceps sinensis mycelium." BIOLOGY OF REPRODUCTION. MAY 2004, vol. 70, no. 5, May 2004 (2004-05), pages 1358-1364, XP002342091 ISSN: 0006-3363</text></B562><B562><text>TAKEUCHI T ET AL: "Effect of traditional herbal medicine, shakuyaku-kanzo-to on total and free serum testosterone levels." THE AMERICAN JOURNAL OF CHINESE MEDICINE. 1989, vol. 17, no. 1-2, 1989, pages 35-44, XP008051240 ISSN: 0192-415X</text></B562><B562><text>OTA H ET AL: "[Stimulatory action of shakuyaku on aromatase activity in cultured rat follicles]" NIPPON SANKA FUJINKA GAKKAI ZASSHI. MAY 1989, vol. 41, no. 5, May 1989 (1989-05), pages 525-529, XP008051238 ISSN: 0300-9165</text></B562><B562><text>TAKAHASHI K ET AL: "Effect of TJ-68 (shakuyaku-kanzo-to) on polycystic ovarian disease." INTERNATIONAL JOURNAL OF FERTILITY AND MENOPAUSAL STUDIES. 1994 MAR-APR, vol. 39, no. 2, March 1994 (1994-03), pages 69-76, XP008051237 ISSN: 1069-3130</text></B562><B562><text>DATABASE BIOSIS [Online] BIOSCIENCES INFORMATION SERVICE, PHILADELPHIA, PA, US; 1982, BELLINO F L ET AL: "ESTROGEN SYNTHETASE STIMULATION BY DI BUTYRYL CYCLIC AMP IN HUMAN CHORIO CARCINOMA CELL CULTURE THE RELATIVE BIOSYNTHETIC RATE OF THE NADP REDUCED FORM CYTOCHROME C REDUCTASE COMPONENT" XP002342115 Database accession no. PREV198375073483 &amp; ENDOCRINOLOGY, vol. 111, no. 4, 1982, pages 1038-1044, ISSN: 0013-7227</text></B562><B562><text>BAIL LE J-C ET AL: "Chalcones are potent inhibitors of aromatase and 17.beta.-hydroxysteroid dehydrogenase activities" LIFE SCIENCES, PERGAMON PRESS, OXFORD, GB, vol. 68, 2001, pages 751-761, XP002241304 ISSN: 0024-3205</text></B562><B562><text>YEH-CHIH KAO ET AL: "MOLECULAR BASIS OF THE INHIBITION OF HUMAN AROMATASE (ESTROGEN SYNTHETASE) BY FLAVONE AND ISOFLAVONE PHYTOESTROGENS: A SITE-DIRECTED MUTAGENESIS STUDY" ENVIRONMENTAL HEALTH PERSPECTIVES, vol. 106, no. 2, February 1998 (1998-02), pages 85-92, XP000981752 ISSN: 0091-6765</text></B562><B562><text>GUTHRIE N ET AL: "EFFECTIVENESS OF CITRUS FLAVONOIDS ON HUMAN PROSTATE, COLON, LUNG, AND MELANOMA CANCER-CELL PROLIFERATION" AMERICAN CHEMICAL SOCIETY. ABSTRACTS OF PAPER. AT THE NATIONAL MEETING, AMERICAN CHEMICAL SOCIETY, WASHINGTON, DC, US, vol. 219, no. 1/2, 26 March 2000 (2000-03-26), page AFGD183, XP008016727 ISSN: 0065-7727</text></B562></B560></B500><B700><B720><B721><snm>Kakuo, Shingo,
c/o Kao Corporation</snm><adr><str>Research Laboratories,
2606, Akabane</str><city>Ichikaimachi,
Haga-gun,
Tochigi 321-3497</city><ctry>JP</ctry></adr></B721><B721><snm>Moriwaki, Shigeru,
c/o Kao Corporation</snm><adr><str>Research Laboratories,
2606, Akabane</str><city>Ichikaimachi,
Haga-gun,
Tochigi 321-3497</city><ctry>JP</ctry></adr></B721><B721><snm>Ohuchi, Atsushi,
c/o Kao Corporation</snm><adr><str>Research Laboratories,
2606, Akabane</str><city>Ichikaimachi,
Haga-gun,
Tochigi 321-3497</city><ctry>JP</ctry></adr></B721><B721><snm>Kusuoku, Hiroshi,
c/o Kao Corporation</snm><adr><str>Research Laboratories,
2606, Akabane</str><city>Ichikaimachi,
Haga-gun,
Tochigi 321-3497</city><ctry>JP</ctry></adr></B721></B720><B730><B731><snm>KAO CORPORATION</snm><iid>100155219</iid><irf>109 251 a/npo</irf><adr><str>14-10, Nihonbashi Kayaba-cho 1-chome, 
Chuo-ku</str><city>Tokyo 103-8210</city><ctry>JP</ctry></adr></B731></B730><B740><B741><snm>Hoffmann Eitle</snm><iid>100061036</iid><adr><str>Patent- und Rechtsanwälte PartmbB 
Arabellastraße 30</str><city>81925 München</city><ctry>DE</ctry></adr></B741></B740></B700><B800><B840><ctry>DE</ctry><ctry>FR</ctry><ctry>GB</ctry></B840><B880><date>20051228</date><bnum>200552</bnum></B880></B800></SDOBI>
</ep-patent-document>
