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<ep-patent-document id="EP04741432B8W1" file="EP04741432W1B8.xml" lang="en" country="EP" doc-number="1608655" kind="B8" correction-code="W1" date-publ="20081015" status="c" dtd-version="ep-patent-document-v1-3">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  2999001/0</B007EP></eptags></B000><B100><B110>1608655</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20081015</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>04741432.1</B210><B220><date>20040322</date></B220><B240><B241><date>20051021</date></B241><B242><date>20070725</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>MI20030573</B310><B320><date>20030324</date></B320><B330><ctry>IT</ctry></B330></B300><B400><B405><date>20081015</date><bnum>200842</bnum></B405><B430><date>20051228</date><bnum>200552</bnum></B430><B450><date>20080716</date><bnum>200829</bnum></B450><B452EP><date>20080121</date></B452EP><B480><date>20081015</date><bnum>200842</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 487/04        20060101AFI20041207BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/4188      20060101ALI20041207BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>PYRROLOIMIDAZOLDERIVATE ,VERFAHERN ZU IHRER HERSTELLUNG, DIESE ENTHALTENDE ZUSAMMENSETZUNGEN, UND IHRE VERWENDUNG ALS NOOTROPIKA</B542><B541>en</B541><B542>PYRROLOIMIDAZOLE DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE  AS NOOTROPIC AGENTS</B542><B541>fr</B541><B542>COMPOSES PRESENTANT UNE ACTION NOOTROPIQUE, LEUR PREPARATION, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, ET LEUR UTILISATION</B542></B540><B560><B561><text>EP-A- 0 174 136</text></B561><B561><text>EP-A- 0 335 483</text></B561><B561><text>WO-A-93/09120</text></B561><B562><text>MARIO PINZA ET AL.: "Synthesis and Pharmacological Activity of a Series of Dihydro-1H-pyrrolo[1,2-a]imidazole-2,5(3H, 6H)-diones, a Novel Class of Potent Cognition Enhancers" JOURNAL OF MEDICINAL CHEMISTRY., vol. 36, no. 26, 24 December 1993 (1993-12-24), pages 4214-4220, XP002295812 USAMERICAN CHEMICAL SOCIETY.</text></B562></B560></B500><B700><B720><B721><snm>FARINA, Carlo
c/o NIKEM RESEARCH S.R.L.</snm><adr><str>Via Zambeletti 25</str><city>I-20021 BARANZATE DI BOLLATE</city><ctry>IT</ctry></adr></B721><B721><snm>GAGLIARDI, Stefania
c/o NIKEM RESEARCH S.R.L.</snm><adr><str>Via Zambeletti 25</str><city>I-20021 BARANZATE DI BOLLATE</city><ctry>IT</ctry></adr></B721><B721><snm>PARINI, Carlo
c/o NIKEM RESEARCH S.R.L.</snm><adr><str>Via Zambeletti 25</str><city>I-20021 BARANZATE DI BOLLATE</city><ctry>IT</ctry></adr></B721><B721><snm>MARTINELLI, Marisa
c/o NIKEM RESEARCH S.R.L.</snm><adr><str>Via Zambeletti 25</str><city>I-20021 BARANZATE DI BOLLATE</city><ctry>IT</ctry></adr></B721><B721><snm>GHELARDINI, Carla;
c/o Dipartimento di</snm><adr><str>Farmacologia Preclinica e Clinica "M. Aiazzi</str><city>Mancini"
Università di Firenze</city><ctry>IT</ctry></adr></B721></B720><B730><B731><snm>BRANE DISCOVERY SRL IN LIQUIDAZIONE</snm><iid>08653350</iid><irf>4050PTEP-CA</irf><adr><str>Via Zambeletti 25</str><city>20021 Baranzate</city><ctry>IT</ctry></adr></B731></B730><B740><B741><snm>Gerli, Paolo</snm><sfx>et al</sfx><iid>00089932</iid><adr><str>Notarbartolo &amp; Gervasi S.p.A. 
Corso di Porta Vittoria, 9</str><city>20122 Milano</city><ctry>IT</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>TR</ctry></B840><B844EP><B845EP><ctry>AL</ctry><date>20051021</date></B845EP><B845EP><ctry>LT</ctry><date>20051021</date></B845EP><B845EP><ctry>LV</ctry><date>20051021</date></B845EP><B845EP><ctry>MK</ctry><date>20051021</date></B845EP></B844EP><B860><B861><dnum><anum>EP2004050339</anum></dnum><date>20040322</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2004085438</pnum></dnum><date>20041007</date><bnum>200441</bnum></B871></B870></B800></SDOBI>
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