(19)
(11) EP 1 644 322 A1

(12)

(43) Date of publication:
12.04.2006 Bulletin 2006/15

(21) Application number: 03796897.1

(22) Date of filing: 10.12.2003
(51) International Patent Classification (IPC): 
C07C 237/22(1990.01)
C07C 237/14(1990.01)
C07D 307/02(1985.01)
C07D 249/08(1985.01)
C07C 311/08(1990.01)
C07D 285/06(1985.01)
A61K 31/166(2000.01)
C07K 5/02(1985.01)
C07C 237/12(1990.01)
C07D 333/02(1985.01)
C07D 211/04(1985.01)
C07C 311/16(1990.01)
C07D 275/02(1985.01)
C07D 213/04(1985.01)
A61P 25/28(2000.01)
C07D 241/08(1985.01)
(86) International application number:
PCT/US2003/039276
(87) International publication number:
WO 2005/005374 (20.01.2005 Gazette 2005/03)
(84) Designated Contracting States:
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR

(30) Priority: 16.06.2003 US 462127
16.06.2003 WO PCT/US03/18858

(71) Applicant: Sunesis Pharmaceuticals, Inc.
San Francisco, CA 94080 (US)

(72) Inventor:
  • YANG, Wenjin
    Foster City, CA 94404 (US)

(74) Representative: Gambell, Derek et al
Graham Watt & Co LLP St Botolph's House 7-9 St Botolph's Road
Sevenoaks Kent TN13 3AJ
Sevenoaks Kent TN13 3AJ (GB)

   


(54) ASPARTYL PROTEASE INHIBITORS